ENSIKLOPEDIA Cari Tekan Enter untuk memulai pencarian cepat. Kembali ke Ensiklopedia Arsip Wikipedia Indonesia Transporter modulator Reuptake modulatorType of pharmaceutical drug This article does not cite any sources. Please help improve this article by adding citations to reliable sources. Unsourced material may be challenged and removed.Find sources: "Reuptake modulator" – news · newspapers · books · scholar · JSTOR (January 2015) (Learn how and when to remove this message) A reuptake modulator, or transporter modulator, is a type of drug which modulates the reuptake of one or more neurotransmitters via their respective neurotransmitter transporters. Examples of reuptake modulators include reuptake inhibitors (transporter blockers) and reuptake enhancers. See also Releasing agent Release modulator Transporter substrate Channel modulator Receptor modulator SSRI vteReceptor/signaling modulatorsAmino acids andsimilar/related Amino acids and related: GABA receptor modulators GABAA receptor positive modulators GABA metabolism and transport modulators GHB receptor modulators Glutamate metabolism and transport modulators Glycine receptor modulators Ionotropic glutamate receptor modulators Metabotropic glutamate receptor modulators Monoamines: Adrenergic receptor modulators Dopamine receptor modulators Histamine receptor modulators Melatonin receptor modulators Monoamine metabolism modulators Monoamine neurotoxins Monoamine releasing agents Monoamine reuptake inhibitors Serotonin receptor modulators hTAAR modulators Acetylcholine: Acetylcholine metabolism and transport modulators Muscarinic acetylcholine receptor modulators Nicotinic acetylcholine receptor modulators Others: Imidazoline receptor modulators Purine receptor modulators Sigma receptor modulators Thyroid hormone receptor modulators Lipids Eicosanoids: Cannabinoid receptor modulators Leukotriene signaling modulators Prostanoid signaling modulators Phospholipids: Lysophospholipid signaling modulators PAF receptor modulators Steroids: Androgen receptor modulators Estrogen receptor modulators Glucocorticoid receptor modulators Mineralocorticoid receptor modulators Progesterone receptor modulators Steroid metabolism modulators Other nuclear receptors: Aryl hydrocarbon receptor modulators Estrogen-related receptor modulators FXR and LXR modulators PPAR modulators Retinoid receptor modulators Vitamin D receptor modulators Xenobiotic-sensing receptor modulators Peptides/proteins Peptides: Angiotensin receptor modulators GH/IGF-1 axis signaling modulators GnRH and gonadotropin receptor modulators Melanocortin receptor modulators Neurokinin receptor modulators Opioid receptor modulators Oxytocin and vasopressin receptor modulators Cytokines: Cytokine receptor modulators Chemokine receptor modulators Interleukin receptor modulators TNF receptor superfamily modulators Growth factors: Growth factor receptor modulators TGFβ receptor superfamily modulators Others andnon-receptor Enzymes: Cytochrome P450 modulators Histone deacetylase inhibitors Phosphodiesterase inhibitors Ion channels: Ion channel modulators TRP channel modulators Transporters: Sodium-glucose transporter modulators Symporter inhibitors Others: Nitric oxide signaling modulators vtePharmacomodulationTypes ♦ Enzyme: Inducer Inhibitor ♦ Ion channel: Opener Blocker ♦ Receptor: Agonist Partial agonist Antagonist Inverse agonist Positive allosteric modulator (PAM) Negative allosteric modulator (NAM) ♦ Transporter [Reuptake vs Efflux]: Enhancer (RE) Inhibitor (RI) Releaser (RA) ♦ Miscellaneous: Precursor Cofactor ClassesEnzymesee Enzyme inhibitionIon channelSee Ion channel modulatorsReceptor &transporterBA/MAdrenergic Adrenergic receptor agonist (α β (1 2)) Adrenergic receptor antagonist (α (1 2) β) Norepinephrine reuptake inhibitor (NRI) Dopaminergic Dopamine receptor agonist Dopamine receptor antagonist Dopamine reuptake inhibitor (DRI) Histaminergic Histamine receptor agonist Histamine receptor antagonist (H1 H2 H3) Serotonergic Serotonin receptor agonist Serotonin receptor antagonist (5-HT3) Serotonin reuptake inhibitor (SRI) AAGABAergic GABA receptor agonist GABA receptor antagonist GABA reuptake inhibitor (GRI) Glutamatergic Glutamate receptor agonist (AMPA) Glutamate receptor antagonist (NMDA) Glutamate reuptake inhibitor Cholinergic Acetylcholine receptor agonist (Muscarinic Nicotinic) Cholinesterase inhibitor Acetylcholine receptor antagonist (Muscarinic Nicotinic (Ganglionic Muscular)) Cannabinoidergic Cannabinoid receptor agonist Cannabinoid receptor antagonist Endocannabinoid enhancer (eCBE) Endocannabinoid reuptake inhibitor (eCBRI) Opioidergic Opioid modulator Opioid receptor agonist Opioid receptor antagonist Enkephalinase inhibitor Other Adenosine reuptake inhibitor (AdoRI) Angiotensin II receptor antagonist Endothelin receptor antagonist NK1 receptor antagonist Vasopressin receptor antagonist Miscellaneous Cofactor (see Enzyme cofactors) Precursor (see Amino acids) This pharmacology-related article is a stub. 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